Tetrahedron letters

A concise synthesis of aza-dipeptide isosteres

A Fässler, G Bold, H Steiner

Index: Faessler, Alex; Bold, Guido; Steiner, Heinz Tetrahedron Letters, 1998 , vol. 39, # 27 p. 4925 - 4928

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Citation Number: 20

Abstract

Download full text in PDF Opens in a new window. Article suggestions will be shown in a dialog on return to ScienceDirect. ... Please enable JavaScript to use all the features on this page. ... Aza-dipeptide isosteres as potent HIV-protease inhibitors containing a (hydroxyethyl)-hydrazine moiety are synthesised in >98% diastereomeric and enantiomeric purity starting from (L)-phenylalanine aldehyde. ... Aza-dipeptide isosteres are synthesised in > 98% de and ee starting from ...

~58%

Process research and development for an efficient synthesis ...

[Xu, Zhongmin; Singh, Janak; Schwinden, Mark D.; Zheng, Bin; Kissick, Thomas P.; Patel, Bharat; Humora, Michael J.; Quiroz, Fernando; Dong, Lin; Hsieh, Dau-Ming; Heikes, James E.; Pudipeddi, Madhusudhan; Lindrud, Mark D.; Srivastava, Sushil K.; Kronenthal, David R.; Mueller, Richard H. Organic Process Research and Development, 2002 , vol. 6, # 3 p. 323 - 328]

New aza-dipeptide analogues as potent and orally absorbed HI...

[Journal of Medicinal Chemistry, , vol. 41, # 18 p. 3387 - 3401]