Angewandte Chemie International Edition

Chemoselective Benzylic C H Activations for the Preparation of Condensed N??Heterocycles

H Ren, P Knochel

Index: Ren, Hongjun; Knochel, Paul Angewandte Chemie - International Edition, 2006 , vol. 45, # 21 p. 3462 - 3465

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Citation Number: 87

Abstract

3463 Angew. Chem. Int. Ed. 2006, 45, 3462–3465 2006 Wiley-VCH Verlag GmbH & Co. KGaA, Weinheim www. angewandte. org cyclization with a CÀH activation, leading to the heterocycles 16 a–c in 74–85% yield and demonstrating the broad scope of this type of ring closure (Scheme 4). In summary, we have reported new Pd-catalyzed cyclizations leading to condensed N-heterocycles. The key step of these ring closures is a chemoselective ...