Antihistamine-1 structure
|
Common Name | Antihistamine-1 | ||
---|---|---|---|---|
CAS Number | 1186430-60-3 | Molecular Weight | 389.47 | |
Density | N/A | Boiling Point | N/A | |
Molecular Formula | C23H24FN5 | Melting Point | N/A | |
MSDS | N/A | Flash Point | N/A |
Use of Antihistamine-1Antihistamine-1 is a H1-antihistamine (Ki=6.9 nM) with acceptable blood-brain barrier penetration and also an inhibitor of CYP2D6 and hERG channel with IC50s of 5.4 and 0.8 μM, respectively. |
Name | Antihistamine-1 |
---|
Description | Antihistamine-1 is a H1-antihistamine (Ki=6.9 nM) with acceptable blood-brain barrier penetration and also an inhibitor of CYP2D6 and hERG channel with IC50s of 5.4 and 0.8 μM, respectively. |
---|---|
Related Catalog | |
Target |
CYP2D6:5.4 μM (IC50) |
In Vitro | Antihistamine-1 (Compound 2) is a H1-antihistamine (Ki=6.9 nM) with acceptable blood-brain barrier penetration and also an inhibitor of CYP2D6 and hERG channel with IC50s of 5.4 and 0.8 μM, respectively[1]. |
References |
Molecular Formula | C23H24FN5 |
---|---|
Molecular Weight | 389.47 |
Storage condition | 2-8℃ |