129173-57-5

129173-57-5 structure

Name: RS-5773
Chemical Name: [(2S,3S)-5-[2-(dimethylamino)ethyl]-2-(4-methoxyphenyl)-4-oxo-8-(thiophen-2-ylmethyl)-2,3-dihydro-1,5-benzothiazepin-3-yl] acetate,hydrochloride
CAS Number: 129173-57-5
Molecular Formula: C₂₇H₃₁ClN₂O₄S₂
Molecular Weight: 547.12900
Catalog: Signaling Pathways Membrane Transporter/Ion Channel Calcium Channel
Create Date: 2016-07-26 23:34:33
Modify Date: 2024-02-29 16:31:52
RS-5773 is a calcium channel inhibitor and a diltiazem congener. RS-5773 has antianginal effect and does not cause excessive hypotension or depression of atrioventricular conduction [1].

Name	[(2S,3S)-5-[2-(dimethylamino)ethyl]-2-(4-methoxyphenyl)-4-oxo-8-(thiophen-2-ylmethyl)-2,3-dihydro-1,5-benzothiazepin-3-yl] acetate,hydrochloride

Description	RS-5773 is a calcium channel inhibitor and a diltiazem congener. RS-5773 has antianginal effect and does not cause excessive hypotension or depression of atrioventricular conduction [1].
Related Catalog	Signaling Pathways >> Membrane Transporter/Ion Channel >> Calcium Channel Research Areas >> Neurological Disease
Target	IC50: Calcium channel[1]
References	[1]. H Shiga, et al. Antianginal effect of RS-5773, a diltiazem congener, in the methacholine-induced anginal model in rats. Jpn J Pharmacol . 1996 Dec;72(4):365-74.