447405-11-0

447405-11-0 structure
447405-11-0 structure
  • Name: FR252384
  • Chemical Name: FR252384
  • CAS Number: 447405-11-0
  • Molecular Formula: C18H17N3
  • Molecular Weight: 275.35
  • Catalog: Signaling Pathways GPCR/G Protein Neuropeptide Y Receptor
  • Create Date: 2018-01-05 13:03:42
  • Modify Date: 2024-01-10 17:42:25
  • FR252384 is a neuropeptide Y-Y5 receptor antagonist, with an IC50 of 2.3 nM.

Name FR252384
Description FR252384 is a neuropeptide Y-Y5 receptor antagonist, with an IC50 of 2.3 nM.
Related Catalog
Target

IC50: 2.3 nM (neuropeptide Y-Y5 receptor)[1]

In Vivo FR252384 is orally absorbable and permeable to brain[1].
References

[1]. Satoh Y, et al. Novel potent antagonists of human neuropeptide Y-Y5 receptor. Part 4: tetrahydrodiazabenzazulene derivatives. Bioorg Med Chem Lett. 2002 Apr 8;12(7):1009-11.

Molecular Formula C18H17N3
Molecular Weight 275.35