934016-19-0
934016-19-0 structure
- Name: Degarelix (acetate)
- Chemical Name: EXT215F4ZU
- CAS Number: 934016-19-0
- Molecular Formula: C84H107ClN18O18
- Molecular Weight: 1692.311
- Create Date: 2018-06-03 07:00:23
- Modify Date: 2025-08-23 13:28:44
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Degarelix is a synthetic gonadotropin-releasing hormone receptor (GNRHR) antagonist (IC50 = 3 nM in HEK293 cells expressing the human receptor).
| Name | EXT215F4ZU |
|---|---|
| Synonyms |
(4S)-N-{4-[(2S,5S,8R,11R,14R)-2-({(2R)-1-{[(2S)-1-{[(2S)-1-[(2S)-2-{[(2R)-1-Amino-1-oxo-2-propanyl]carbamoyl}-1-pyrrolidinyl]-6-(isopropylamino)-1-oxo-2-hexanyl]amino}-4-methyl-1-oxo-2-pentanyl]amino}-3-[4-(carbamoylamino)phenyl]-1-oxo-2-propanyl}carbamoyl)-11-(4-chlorobenzyl)-5-(hydroxymethyl)-14-(2-naphthylmethyl)-4,7,10,13,16-pentaoxo-8-(3-pyridinylmethyl)-3,6,9,12,15-pentaazaheptadec-1-yl]phenyl}-2,6-dioxohexahydro-4-pyrimidinecarboxami
EXT215F4ZU |
| Molecular Formula | C84H107ClN18O18 |
|---|---|
| Molecular Weight | 1692.311 |
| Exact Mass | 1690.769897 |