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2138814-32-9

2138814-32-9 structure
2138814-32-9 structure
  • Name: GSK3004774
  • Chemical Name: GSK3004774
  • CAS Number: 2138814-32-9
  • Molecular Formula: C32H40N4O3
  • Molecular Weight: 528.69
  • Catalog: Signaling Pathways GPCR/G Protein CaSR
  • Create Date: 2019-03-03 11:40:15
  • Modify Date: 2024-01-11 17:20:46
  • GSK3004774 is a potent, nonabsorbable agonist of CaSR, with an pEC50 of 7.3, 6.6 and 6.5 for human, mouse and rat CaSR, respectively. GSK3004774 shows an EC50 of 50 nM for human CaSR[1].

Name GSK3004774
Description GSK3004774 is a potent, nonabsorbable agonist of CaSR, with an pEC50 of 7.3, 6.6 and 6.5 for human, mouse and rat CaSR, respectively. GSK3004774 shows an EC50 of 50 nM for human CaSR[1].
Related Catalog
References

[1]. Sparks SM, et al. Identification of potent, nonabsorbable agonists of the calcium-sensing receptor for GI-specific administration. Bioorg Med Chem Lett. 2017 Oct 15;27(20):4673-4677.

Molecular Formula C32H40N4O3
Molecular Weight 528.69