1176326-76-3

1176326-76-3 structure
1176326-76-3 structure
  • Name: DSP-1053
  • Chemical Name: DSP-1053
  • CAS Number: 1176326-76-3
  • Molecular Formula: C26H32BrNO4
  • Molecular Weight: 502.44
  • Catalog: Signaling Pathways Neuronal Signaling Serotonin Transporter
  • Create Date: 2019-03-31 09:23:33
  • Modify Date: 2024-01-20 19:38:33
  • DSP-1053 is a potent Serotonin Transporter (SERT) (Ki=1.02 nM) inhibitor with partial 5-HT1A receptor (Ki=5.05 nM) agonistic activity.

Name DSP-1053
Description DSP-1053 is a potent Serotonin Transporter (SERT) (Ki=1.02 nM) inhibitor with partial 5-HT1A receptor (Ki=5.05 nM) agonistic activity.
Related Catalog
Target

Ki: 1.02 nM (SERT), 1.02 nM (5-HT1A)[1]

References

[1]. Yoshinaga H, et al. Discovery of DSP-1053, a novel benzylpiperidine derivative with potent serotonin transporter inhibitory activity and partial 5-HT1A receptor agonistic activity. Bioorg Med Chem. 2018 May 1;26(8):1614-1627.

Molecular Formula C26H32BrNO4
Molecular Weight 502.44
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