DC Chemicals Limited
China
Product Name: San78-130
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Purity: 98.0%
Stocking Period: 3 Day
Contact: Tony Cao

66018-45-9

66018-45-9 structure

66018-45-9 structure

Name: San78-130
Chemical Name: San78-130
CAS Number: 66018-45-9
Molecular Formula: C₁₉H₂₆O₇
Molecular Weight: 366.41
Catalog: Research Areas Cancer
Create Date: 2019-08-04 09:50:59
Modify Date: 2024-01-24 17:48:37
San78-130 is a selective and potent ALK1 inhibitor with an IC50 of 62 nM. San78-130 also inhibits FLT4/VEGFR3, KDR/VEGFR2, MEK2, and FLT3 with IC50s of 114, 162, 186.7, and 188 nM, respectively[1].

Name	San78-130

Description	San78-130 is a selective and potent ALK1 inhibitor with an IC50 of 62 nM. San78-130 also inhibits FLT4/VEGFR3, KDR/VEGFR2, MEK2, and FLT3 with IC50s of 114, 162, 186.7, and 188 nM, respectively[1].
Related Catalog	Research Areas >> Cancer
Target	ALK1:62 nM (IC50) FLT4/VEGFR3:114 nM (IC50) KDR/VEGFR2:162 nM (IC50) MEK2:186.7 nM (IC50) FLT3:188 nM (IC50)
References	[1]. Cho H, et al. Identification of the First Selective Activin Receptor-Like Kinase 1 Inhibitor, a Reversible Version of L-783277. J Med Chem. 2017 Feb 23;60(4):1495-1508.

Molecular Formula	C₁₉H₂₆O₇
Molecular Weight	366.41