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1998139-29-9

1998139-29-9 structure
1998139-29-9 structure
  • Name: MMSET-IN-1
  • Chemical Name: MMSET-IN-1
  • CAS Number: 1998139-29-9
  • Molecular Formula: C18H29N7O5
  • Molecular Weight: 423.47
  • Catalog: Research Areas Cancer
  • Create Date: 2019-09-09 11:09:50
  • Modify Date: 2025-09-01 22:35:15
  • MMSET-IN-1 is a multiple myeloma SET domain (MMSET, aka NSD2/WHSC1) inhibitor against SETD2 and MMSET with IC50s of 0.49 and 3.3 μM, respectively. MMSET-IN-1 has a Kd of 1.6 μM for MMSET[1].

Name MMSET-IN-1
Description MMSET-IN-1 is a multiple myeloma SET domain (MMSET, aka NSD2/WHSC1) inhibitor against SETD2 and MMSET with IC50s of 0.49 and 3.3 μM, respectively. MMSET-IN-1 has a Kd of 1.6 μM for MMSET[1].
Related Catalog
Target

IC50: 0.49 μM (SETD2), 3.3 μM (MMSET)[1] Kd: 1.6 μM[1]

References

[1]. Tisi D, et al. Structure of the Epigenetic Oncogene MMSET and Inhibition by N-Alkyl Sinefungin Derivatives. ACS Chem Biol. 2016 Nov 18;11(11):3093-3105.

Molecular Formula C18H29N7O5
Molecular Weight 423.47
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