1627136-55-3
1627136-55-3 structure
- Name: RSK2-IN-20
- Chemical Name: RSK2-IN-20
- CAS Number: 1627136-55-3
- Molecular Formula: C21H18N6O3
- Molecular Weight: 402.414
- Create Date: 2020-01-12 20:37:27
- Modify Date: 2024-09-23 18:05:27
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RSK2-IN-20 is a potent, selective, and durable inhibitpr of RSK2 with IC50 of 47 nM; shows high selectivity over NEK2, PLK1; potently inhibits MSK1 autophosphorylation in cells, and has no significant effect on a panel of 18 additional kinases.
| Name | RSK2-IN-20 |
|---|
| Description | RSK2-IN-20 is a potent, selective, and durable inhibitpr of RSK2 with IC50 of 47 nM; shows high selectivity over NEK2, PLK1; potently inhibits MSK1 autophosphorylation in cells, and has no significant effect on a panel of 18 additional kinases. |
|---|---|
| References | References 1. Krishnan S, et al. J Am Chem Soc. 2014 Sep 10;136(36):12624-30. View Related Products by Target Ribosomal S6 Kinase (RSK) |
| Molecular Formula | C21H18N6O3 |
|---|---|
| Molecular Weight | 402.414 |