616884-67-4

616884-67-4 structure
616884-67-4 structure
  • Name: OMDM-6
  • Chemical Name: OMDM-6
  • CAS Number: 616884-67-4
  • Molecular Formula: C28H42N2O3
  • Molecular Weight: 454.64
  • Catalog: Signaling Pathways GPCR/G Protein Cannabinoid Receptor
  • Create Date: 2020-06-01 13:51:11
  • Modify Date: 2025-08-20 11:07:00
  • OMDM-6 is a hybrid agonist of vanilloid receptor type 1 (VR1, TRPV1) (EC50=75 nM) and cannabinoid receptor type 1 (CB1) (Ki=3.2 μM). OMDM-6 inhibits anandamide cellular uptake (ACU) with a Ki of 7.0 μM[1].

Name OMDM-6
Description OMDM-6 is a hybrid agonist of vanilloid receptor type 1 (VR1, TRPV1) (EC50=75 nM) and cannabinoid receptor type 1 (CB1) (Ki=3.2 μM). OMDM-6 inhibits anandamide cellular uptake (ACU) with a Ki of 7.0 μM[1].
Related Catalog
Target

EC50: 75 nM (vanilloid receptor type 1), Ki: 3.2 μM (cannabinoid receptor type 1), Ki: 7.0 μM (anandamide cellular uptake)[1]

References

[1]. Ortar G, et al. Novel selective and metabolically stable inhibitors of anandamide cellular uptake. Biochem Pharmacol. 2003 May 1;65(9):1473-81.

Molecular Formula C28H42N2O3
Molecular Weight 454.64
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