782485-03-4

782485-03-4 structure

Name: [Orn5]-URP TFA
Chemical Name: [Orn5]-URP
CAS Number: 782485-03-4
Molecular Formula: C₄₈H₆₂N₁₀O₁₀S₂
Molecular Weight: 1003.20
Catalog: Signaling Pathways GPCR/G Protein Urotensin Receptor
Create Date: 2020-08-09 12:37:09
Modify Date: 2024-01-08 23:44:45
[Orn5]-URP is a potent and selective pure antagonist of Urotensin-II receptor (UT), with an pEC50 of 7.24. [Orn5]-URP displays no agonist activity[1][2].

Name	[Orn5]-URP

Description	[Orn5]-URP is a potent and selective pure antagonist of Urotensin-II receptor (UT), with an pEC50 of 7.24. [Orn5]-URP displays no agonist activity[1][2].
Related Catalog	Research Areas >> Cardiovascular Disease Signaling Pathways >> GPCR/G Protein >> Urotensin Receptor
Target	pEC50: 7.24[2]
References	[1]. Diallo M, et, al. [Orn5]URP acts as a pure antagonist of urotensinergic receptors in rat cortical astrocytes. Peptides. 2008 May; 29(5): 813-9. [2]. David C, et, al. Structure-activity relationships and structural conformation of a novel urotensin II-related peptide. Peptides. 2004 Oct; 25(10): 1819-30.