Shanghai Nianxing Industrial Co., Ltd
China
Product Name: GPR30 agonist-1
Price:
Purity: 98.0%
Stocking Period: 10 Day
Contact: Yang

DC Chemicals Limited
China
Product Name: GPR30 agonist-1
Price: ￥Inquiry/1g
Purity: 98.9%
Stocking Period: 1 Day
Contact: Tony Cao

415919-74-3

415919-74-3 structure

415919-74-3 structure

Name: GPR30 agonist-1
Chemical Name: GPR30 agonist-1
CAS Number: 415919-74-3
Molecular Formula: C₁₉H₁₇BrFNO
Molecular Weight: 374.25
Catalog: Research Areas Cardiovascular Disease
Create Date: 2021-09-10 20:20:40
Modify Date: 2024-01-09 12:06:00
GPR30 agonist-1 is a G protein-coupled receptor 30 (GPR30) agonist. GPR30 agonist-1 exerts vasorelaxant effects[1].

Name	GPR30 agonist-1

Description	GPR30 agonist-1 is a G protein-coupled receptor 30 (GPR30) agonist. GPR30 agonist-1 exerts vasorelaxant effects[1].
Related Catalog	Signaling Pathways >> Others >> Estrogen Receptor/ERR Research Areas >> Cardiovascular Disease Research Areas >> Endocrinology
In Vivo	GPR30 agonist-1 (compound 5408-0877) (1 nM-10 μM) induces a concentration-dependent relaxation in carotid arteries from both male and female rats. GPR30 agonist-1-induced relaxation is abolished by endothelium removal and abrogated in the presence of the nitric oxide synthase inhibitor NG-nitro-l-arginine methyl ester (100 μM)[1].
References	[1]. Brad R S Broughton, et al. Endothelium-dependent relaxation by G protein-coupled receptor 30 agonists in rat carotid arteries. Am J Physiol Heart Circ Physiol. 2010 Mar;298(3):H1055-61.

Molecular Formula	C₁₉H₁₇BrFNO
Molecular Weight	374.25