415919-74-3

415919-74-3 structure
415919-74-3 structure
  • Name: GPR30 agonist-1
  • Chemical Name: GPR30 agonist-1
  • CAS Number: 415919-74-3
  • Molecular Formula: C19H17BrFNO
  • Molecular Weight: 374.25
  • Catalog: Research Areas Cardiovascular Disease
  • Create Date: 2021-09-10 20:20:40
  • Modify Date: 2024-01-09 12:06:00
  • GPR30 agonist-1 is a G protein-coupled receptor 30 (GPR30) agonist. GPR30 agonist-1 exerts vasorelaxant effects[1].

Name GPR30 agonist-1
Description GPR30 agonist-1 is a G protein-coupled receptor 30 (GPR30) agonist. GPR30 agonist-1 exerts vasorelaxant effects[1].
Related Catalog
In Vivo GPR30 agonist-1 (compound 5408-0877) (1 nM-10 μM) induces a concentration-dependent relaxation in carotid arteries from both male and female rats. GPR30 agonist-1-induced relaxation is abolished by endothelium removal and abrogated in the presence of the nitric oxide synthase inhibitor NG-nitro-l-arginine methyl ester (100 μM)[1].
References

[1]. Brad R S Broughton, et al. Endothelium-dependent relaxation by G protein-coupled receptor 30 agonists in rat carotid arteries. Am J Physiol Heart Circ Physiol. 2010 Mar;298(3):H1055-61.

Molecular Formula C19H17BrFNO
Molecular Weight 374.25
The content on this webpage is sourced from various professional data sources. If you have any questions or concerns regarding the content, please feel free to contact service1@chemsrc.com.