Name | Adenosine receptor antagonist 1 |
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Description | Adenosine receptor antagonist 1 is a A2aR-selective antagonist with an IC50 of 0.29 nM and displays 14-fold more selective for A2aRthan A2bR. |
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Related Catalog | |
Target |
A2AR:0.29 nM (IC50) |
References |
[1]. Lamb ML, et al. Triazole compounds as adenosine receptor antagonists. WO2021156439A1. |
Molecular Formula | C22H15ClFN7O |
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Molecular Weight | 447.85 |