| Name | EP4 receptor antagonist 4 |
|---|
| Description | EP4 receptor antagonist 4 is an EP4 receptor agonist with the human pEC50 value of 6.3[1]. |
|---|---|
| Related Catalog | |
| Target |
EP4:6.3 (pEC50) |
| In Vitro | EP4 receptor antagonist 4 (24 h) treatment shows agonism in HEK293 cells stably transfected with hEP4[1]. EP4 receptor antagonist 4 (30 min) treatment shows agonism (pEC50<5) and antagonism (pIC50<5)[1]. Cell Viability Assay[1] Cell Line: HEK293 cells Concentration: Incubation Time: 24 hours Result: Exhibited the human pEC50 value of 6.3. |
| References |
[1]. Joannes Theodorus Maria Linders, et al. Bicyclic derivatives as ep4 agonists. WO2008092860A1 |
| Molecular Formula | C19H14N2OS |
|---|---|
| Molecular Weight | 318.39 |