| Name | Cavα2δ1&NET-IN-3 |
|---|
| Description | Cavα2δ1&NET-IN-3 (example 216) is an inhibitor of the subunit α2δ of voltage-gated calcium channels (VGCC) and noradrenaline transporter (NET). Cavα2δ1&NET-IN-3 has Kis of 100-500 nM for human α2δ-1 subunit of Cav2.2 calcium channel and NET, respectively[1]. |
|---|---|
| Related Catalog | |
| Target |
Calcium Channel |
| References |
| Molecular Formula | C24H30N6O2S |
|---|---|
| Molecular Weight | 466.60 |