| Name | LY-466195 |
|---|---|
| Synonyms |
LY466195
3-Isoquinolinecboxylic acid, 6-[[(2S)-2-cboxy-4,4-difluoro-1-pyrrolidinyl]methyl]decahydro-, (3S,4,6S,8) LY466195,LY |
| Description | LY-466195 is a competitive antagonist of GLUK5 receptor. |
|---|---|
| References | 1. Andreou AP, Holland PR, Lasalandra MP, Goadsby PJ. Modulation of nociceptive dural input to the trigeminocervical complex through GluK1 kainate receptors. Pain. 2015 Mar;156(3):439-50. doi: 10.1097/01.j.pain.0000460325.25762.c0. PubMed PMID: 25679470. |
| Molecular Formula | C16H24F2N2O4 |
|---|---|
| Molecular Weight | 346.37 |