157097-10-4

157097-10-4 structure

Name: RLH-033
Chemical Name: 2-(4-phenylpiperidin-1-yl)ethyl 1-(4-nitrophenyl)cyclopentane-1-carboxylate,hydrochloride
CAS Number: 157097-10-4
Molecular Formula: C₂₅H₃₁ClN₂O₄
Molecular Weight: 458.97800
Catalog: Signaling Pathways GPCR/G Protein mAChR
Create Date: 2017-06-21 06:18:25
Modify Date: 2024-04-03 13:00:25
RLH-033 is a potent and selective ligand for the sigma 1 recognition site. RLH-033 has high affinity for sigma 1 sites labeled by [3H](+)-pentazocine with a Ki of 50 pM[1].

Name	2-(4-phenylpiperidin-1-yl)ethyl 1-(4-nitrophenyl)cyclopentane-1-carboxylate,hydrochloride
Synonyms	2-(4-phenylpiperidin-1-yl)ethyl 1-(4-nitrophenyl)cyclopentane-1-carboxylate hydrochloride 2-(4-Phenylpiperidinyl)ethyl 1-(4-nitrophenyl)cyclopentanecarboxylate hydrochloride Rlh 033

Description	RLH-033 is a potent and selective ligand for the sigma 1 recognition site. RLH-033 has high affinity for sigma 1 sites labeled by [3H](+)-pentazocine with a Ki of 50 pM[1].
Related Catalog	Signaling Pathways >> Neuronal Signaling >> mAChR Signaling Pathways >> GPCR/G Protein >> mAChR Research Areas >> Neurological Disease
References	[1]. R L Hudkins, et al. RLH-033, a novel, potent and selective ligand for the sigma 1 recognition site. Eur J Pharmacol. 1994 Dec 12;271(1):235-6.