ORL1 antagonist 2

Modify Date: 2026-04-20 20:18:13

ORL1 antagonist 2 structure	Common Name	ORL1 antagonist 2
	CAS Number	1169982-72-2	Molecular Weight	462.0
	Density	N/A	Boiling Point	N/A
	Molecular Formula	C₂₃H₃₂ClN₅O₃	Melting Point	N/A
	MSDS	N/A	Flash Point	N/A

Name	ORL1 antagonist 2

Molecular Formula	C₂₃H₃₂ClN₅O₃
Molecular Weight	462.0
InChIKey	JSDMNVWPECZJKQ-UHFFFAOYSA-N
SMILES	CCN1CCN(CC1)C2=C(C=C3C(=C2)N=C(N3)C(=O)C4(CCC(CC4)NC(=O)OC)C)Cl

Name: Effect on mouse pgp-mediated efflux assessed as ratio of apparent permeability from a...
Source: ChEMBL
Target: N/A
External Id: CHEMBL1014961

Name: Effect on human pgp-mediated efflux assessed as ratio of apparent permeability from a...
Source: ChEMBL
Target: N/A
External Id: CHEMBL1014960

Name: Displacement of [35S]MK499 from human ERG expressed in HEK293 cells
Source: ChEMBL
Target: Potassium voltage-gated channel subfamily H member 2
External Id: CHEMBL1014963

Name: Antagonist activity against ORL1 receptor by [S35]GTPgammaS binding
Source: ChEMBL
Target: Nociceptin receptor
External Id: CHEMBL1014962

Name: hERG Radioligand Binding Assay from Article 10.1016/j.bmcl.2009.04.023: "2-Cyclohexyl...
Source: BindingDB
Target: N/A
External Id: BindingDB_3257_3

Name: In Vitro Binding Assay (IC50) and In Vitro Agonism/Antagonism Measurements (EC50/IC50...
Source: BindingDB
Target: N/A
External Id: BindingDB_3257_1

Name: Displacement of [125I]Tyr14-NC/OFQ from ORL1 receptor
Source: ChEMBL
Target: Nociceptin receptor
External Id: CHEMBL1012389

Name: Metabolic stability in human liver microsomes assessed as parent compound remaining a...
Source: ChEMBL
Target: Liver microsomes
External Id: CHEMBL1014965

Name: Distribution coefficient, log D at pH 7.4 by shake flask method
Source: ChEMBL
Target: N/A
External Id: CHEMBL1014964

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ORL1 antagonist 2

Names

Chemical & Physical Properties

ORL1 antagonist 2Bioassay

The content on this webpage is sourced from various professional data sources. If you have any questions or concerns regarding the content, please feel free to contact service1@chemsrc.com.