Odapipam structure
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Common Name | Odapipam | ||
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CAS Number | 131796-63-9 | Molecular Weight | 329.82100 | |
Density | 1.269g/cm3 | Boiling Point | 460.4ºC at 760mmHg | |
Molecular Formula | C19H20ClNO2 | Melting Point | N/A | |
MSDS | N/A | Flash Point | 232.2ºC |
Use of OdapipamOdapipam (NNC 756) is a selective, high affinity and benzazepine dopamine D1 receptor antagonist with a Kd of 0.18 nM. Odapipam is also a superior positron emission tomography (PET) radiotracer[1][2]. |
Name | (5S)-8-chloro-5-(2,3-dihydro-1-benzofuran-7-yl)-3-methyl-1,2,4,5-tetrahydro-3-benzazepin-7-ol |
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Synonym | More Synonyms |
Description | Odapipam (NNC 756) is a selective, high affinity and benzazepine dopamine D1 receptor antagonist with a Kd of 0.18 nM. Odapipam is also a superior positron emission tomography (PET) radiotracer[1][2]. |
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Related Catalog | |
Target |
Dopamine D1 receptor[1] |
In Vivo | The metabolism of Odapipam has been studied with phenobarbital-induced rat liver microsomes. During the incubation of Odapipam, five different metabolites are formed. The electron-ionization (EI+) mass spectra of the metabolites indicated the formation of N-desmethyl-Odapipam, 1-hydroxy-Odapipam, the two isomers of 3′-hydroxy-Odapipam and a metabolite which is dehydrogenated in the dihydrobenzofuran moiety[3]. |
References |
Density | 1.269g/cm3 |
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Boiling Point | 460.4ºC at 760mmHg |
Molecular Formula | C19H20ClNO2 |
Molecular Weight | 329.82100 |
Flash Point | 232.2ºC |
Exact Mass | 329.11800 |
PSA | 32.70000 |
LogP | 3.53820 |
Vapour Pressure | 4.27E-09mmHg at 25°C |
Index of Refraction | 1.623 |
HS Code | 2934999090 |
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HS Code | 2934999090 |
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Summary | 2934999090. other heterocyclic compounds. VAT:17.0%. Tax rebate rate:13.0%. . MFN tariff:6.5%. General tariff:20.0% |
Odapipam |
Nnc 756 |
UNII-847PQF7ZN6 |