DKR-1051
Modify Date: 2024-09-13 13:00:19
DKR-1051 structure
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Common Name | DKR-1051 | ||
|---|---|---|---|---|
| CAS Number | 2089053-14-3 | Molecular Weight | 385.474 | |
| Density | N/A | Boiling Point | N/A | |
| Molecular Formula | C24H26F3N | Melting Point | N/A | |
| MSDS | N/A | Flash Point | N/A | |
Use of DKR-1051A novel potent, subtype-selective sigma 2 receptor/PGRMC1 ligand with Ki of 61 nM, 9-fold selectivity over sigma 1 receptors (Ki=556 nM); modulates intracellular Ca2+ levels in human SK-N-SH neuroblastoma cells, relieves spared nerve injury-induced mechanical hypersensitivity in vivo. |
| Name | DKR-1051 |
|---|
| Description | A novel potent, subtype-selective sigma 2 receptor/PGRMC1 ligand with Ki of 61 nM, 9-fold selectivity over sigma 1 receptors (Ki=556 nM); modulates intracellular Ca2+ levels in human SK-N-SH neuroblastoma cells, relieves spared nerve injury-induced mechanical hypersensitivity in vivo. |
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| References | References 1. Yi B, et al. J Neurochem. 2017 Feb;140(4):561-575. 2. Sahn JJ, et al. ACS Chem Neurosci. 2017 Aug 16;8(8):1801-1811. View Related Products by Target Sigma Receptor |
| Molecular Formula | C24H26F3N |
|---|---|
| Molecular Weight | 385.474 |
- Shanghai Nianxing Industrial Co., Ltd
- China
- Product Name: DKR-1051
- Price: ￥Inquiry/100mg ￥Inquiry/250mg ￥Inquiry/500mg
- Purity: 98.0%
- Delivery: 10 Day
- Contact: Huang
- Email: sales@echemcloud.com
- ShangHai DC Chemicals Co.,Ltd
- China
- Product Name: DKR-1051
- Price: ￥Inquiry/1g
- Purity: 98.9%
- Delivery: 1 Day
- Contact: Tony Lai
- Email: order@dcchemicals.com
- DC Chemicals Limited
- China
- Product Name: DKR-1051
- Price: $Inquiry/100mg $Inquiry/250mg $Inquiry/500mg
- Purity: 98.0%
- Delivery: 3 Day
- Contact: Tony Cao
- Email: sales@dcchemicals.com
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