JAK3 covalent inhibitor-1 structure
|
Common Name | JAK3 covalent inhibitor-1 | ||
---|---|---|---|---|
CAS Number | 2300106-50-5 | Molecular Weight | 448.47 | |
Density | N/A | Boiling Point | N/A | |
Molecular Formula | C22H17FN6O2S | Melting Point | N/A | |
MSDS | N/A | Flash Point | N/A |
Use of JAK3 covalent inhibitor-1JAK3 covalent inhibitor-1 is a potent and selective janus kinase 3 (JAK3) covalent inhibitor with an IC50 of 11 nM and shows 246-fold selectivity vs other JAKs[1]. |
Name | JAK3 covalent inhibitor-1 |
---|
Description | JAK3 covalent inhibitor-1 is a potent and selective janus kinase 3 (JAK3) covalent inhibitor with an IC50 of 11 nM and shows 246-fold selectivity vs other JAKs[1]. |
---|---|
Related Catalog | |
Target |
JAK3:11 nM (IC50) |
References |
Molecular Formula | C22H17FN6O2S |
---|---|
Molecular Weight | 448.47 |