5-HT6/5-HT2A receptor ligand-1

Modify Date: 2024-01-06 17:04:07

5-HT6/5-HT2A receptor ligand-1 structure	Common Name	5-HT6/5-HT2A receptor ligand-1
	CAS Number	2411088-07-6	Molecular Weight	350.39
	Density	N/A	Boiling Point	N/A
	Molecular Formula	C₂₁H₁₉FN₂O₂	Melting Point	N/A
	MSDS	N/A	Flash Point	N/A

Use of 5-HT6/5-HT2A receptor ligand-1

5-HT6/5-HT2A receptor ligand-1 (compound 33) is a dual 5-HT6/5-HT2A receptor antagonist, with a Ki of 2 nM and 11 nM, respectively. 5-HT6/5-HT2A receptor ligand-1 has the potential for neurological and psychiatric disorders research[1].

Name	5-HT6/5-HT2A receptor ligand-1

Description	5-HT6/5-HT2A receptor ligand-1 (compound 33) is a dual 5-HT6/5-HT2A receptor antagonist, with a Ki of 2 nM and 11 nM, respectively. 5-HT6/5-HT2A receptor ligand-1 has the potential for neurological and psychiatric disorders research[1].
Related Catalog	Research Areas >> Neurological Disease Signaling Pathways >> GPCR/G Protein >> 5-HT Receptor Signaling Pathways >> Neuronal Signaling >> 5-HT Receptor
Target	5-HT6 Receptor:2 nM (Ki) 5-HT2A Receptor:11 nM (IC50)
References	[1]. Staroń J, et, al. Virtual screening-driven discovery of dual 5-HT 6/5-HT 2A receptor ligands with pro-cognitive properties. Eur J Med Chem. 2020 Jan 1;185:111857.

Molecular Formula	C₂₁H₁₉FN₂O₂
Molecular Weight	350.39

5-HT6/5-HT2A receptor ligand-1

Use of 5-HT6/5-HT2A receptor ligand-1

Names

5-HT6/5-HT2A receptor ligand-1 Biological Activity

Chemical & Physical Properties