ABCG2-IN-1
Modify Date: 2025-09-12 11:19:32
ABCG2-IN-1 structure
|
Common Name | ABCG2-IN-1 | ||
|---|---|---|---|---|
| CAS Number | 2559759-40-7 | Molecular Weight | 468.59 | |
| Density | N/A | Boiling Point | N/A | |
| Molecular Formula | C26H36N4O4 | Melting Point | N/A | |
| MSDS | N/A | Flash Point | N/A | |
Use of ABCG2-IN-1ABCG2-IN-1 (compound K2), a Ko143 analog, is an orally active ABCG2 inhibitor with an IC50 of 0.13 μM. ABCG2-IN-1 has favorable oral pharmacokinetic profiles in mice[1]. |
| Name | ABCG2-IN-1 |
|---|
| Description | ABCG2-IN-1 (compound K2), a Ko143 analog, is an orally active ABCG2 inhibitor with an IC50 of 0.13 μM. ABCG2-IN-1 has favorable oral pharmacokinetic profiles in mice[1]. |
|---|---|
| Related Catalog | |
| Target |
IC50: 0.13 μM (ABCG2)[1] |
| References |
| Molecular Formula | C26H36N4O4 |
|---|---|
| Molecular Weight | 468.59 |
| InChIKey | MJLGVXCTSMTDEP-JBACZVJFSA-N |
| SMILES | COc1ccc2c3c([nH]c2c1)C(CC(C)C)N1C(=O)C(CCC(=O)NC(C)(C)C)NC(=O)C1C3 |