Leucettinib-92
Modify Date: 2024-01-14 21:16:51
Leucettinib-92 structure
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Common Name | Leucettinib-92 | ||
|---|---|---|---|---|
| CAS Number | 2732859-57-1 | Molecular Weight | 378.49 | |
| Density | N/A | Boiling Point | N/A | |
| Molecular Formula | C21H22N4OS | Melting Point | N/A | |
| MSDS | N/A | Flash Point | N/A | |
Use of Leucettinib-92Leucettinib-92 (compound 92) is an inhibitor of DYRK/CLK kinase, The IC50s are 147 nM (CLK1), 39 nM (CLK2), 5.2 nM (CLK4), 0.8 μM (CLK3), 124 nM (DYRK1A), 204 nM (DYRK1B), 0.16 μM (DYRK2), respectively. 1.0 μM (DYRK3), 0.52 μM (DYRK4), 2.78 μM (GSK3)[1]. |
| Name | Leucettinib-92 |
|---|
| Description | Leucettinib-92 (compound 92) is an inhibitor of DYRK/CLK kinase, The IC50s are 147 nM (CLK1), 39 nM (CLK2), 5.2 nM (CLK4), 0.8 μM (CLK3), 124 nM (DYRK1A), 204 nM (DYRK1B), 0.16 μM (DYRK2), respectively. 1.0 μM (DYRK3), 0.52 μM (DYRK4), 2.78 μM (GSK3)[1]. |
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| Related Catalog | |
| Target |
IC50: 147 nM (CLK1), 39 nM (CLK2), 5.2 nM (CLK4), 0.8 μM (CLK3), 124 nM (DYRK1A), 204 nM (DYRK1B), 0.16 μM (DYRK2), 1.0 μM (DYRK3), 0.52 μM (DYRK4), 2.78 μM (GSK3)[1] |
| References |
| Molecular Formula | C21H22N4OS |
|---|---|
| Molecular Weight | 378.49 |