GSK217
Modify Date: 2024-04-09 11:59:35
GSK217 structure
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Common Name | GSK217 | ||
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| CAS Number | 2748687-92-3 | Molecular Weight | 360.421 | |
| Density | N/A | Boiling Point | N/A | |
| Molecular Formula | C20H20N6O | Melting Point | N/A | |
| MSDS | N/A | Flash Point | N/A | |
Use of GSK217GSK217 (GSK-217) is a potent, highly selective BET BD2 inhibitor with pIC50 of 7.5 (BRD4 BD2), 300-fold selectivity over BRD4 BD1. |
| Name | GSK217 |
|---|
| Description | GSK217 (GSK-217) is a potent, highly selective BET BD2 inhibitor with pIC50 of 7.5 (BRD4 BD2), 300-fold selectivity over BRD4 BD1. |
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| References | 1. Helen E Aylott, et al. J Med Chem. 2021 Mar 25;64(6):3249-3281. |
| Molecular Formula | C20H20N6O |
|---|---|
| Molecular Weight | 360.421 |
| InChIKey | MMMRGZLSUKMQOD-UHFFFAOYSA-N |
| SMILES | CCNC(=O)c1cc(Cc2cccc3[nH]ccc23)nc(-c2cn(C)nn2)c1 |