GLUT1-IN-2

Modify Date: 2025-11-21 09:35:20

GLUT1-IN-2 Structure
GLUT1-IN-2 structure
Common Name GLUT1-IN-2
CAS Number 305357-89-5 Molecular Weight 327.38
Density N/A Boiling Point N/A
Molecular Formula C21H17N3O Melting Point N/A
MSDS N/A Flash Point N/A

 Use of GLUT1-IN-2


GLUT1-IN-2 (compound 17) is a GLUT1 inhibitor with an IC50 value of 12 μM. GLUT1-IN-2 shows inhibitory effect to Plasmodium falciparum hexose transporter PfHT with an IC50 value of 13 μM. GLUT1-IN-2 can be used for the research of infection[1].

 Names

Name Benzamide, N-[3-(1H-benzimidazol-2-yl)phenyl]-3-methyl

 GLUT1-IN-2 Biological Activity

Description GLUT1-IN-2 (compound 17) is a GLUT1 inhibitor with an IC50 value of 12 μM. GLUT1-IN-2 shows inhibitory effect to Plasmodium falciparum hexose transporter PfHT with an IC50 value of 13 μM. GLUT1-IN-2 can be used for the research of infection[1].
Related Catalog
Target

IC50: 12 μM (GLUT1), 13 μM (PfHT)[1]

In Vitro GLUT1-IN-2 (0-100 μM) inhibits activities of GLUT1 and PfHT with IC50 values of 12 and 13 μM, respectively[1].

 Chemical & Physical Properties

Molecular Formula C21H17N3O
Molecular Weight 327.38
InChIKey BFAZKDZNMRHORZ-UHFFFAOYSA-N
SMILES Cc1cccc(C(=O)Nc2cccc(-c3nc4ccccc4[nH]3)c2)c1

 GLUT1-IN-2Bioassay

View more

Name: Antileishmanial activity against axenic amastigote Leishmania donovani MHOM/SD/1962/1...
Source: ChEMBL
Target: Leishmania donovani
External Id: CHEMBL3406137
Name: Antileishmanial activity against axenic amastigote Leishmania donovani MHOM/SD/1962/1...
Source: ChEMBL
Target: Leishmania donovani
External Id: CHEMBL3406135
Name: Antibacterial activity against Chlamydia pneumoniae CWL029 infected in human HL cells...
Source: ChEMBL
Target: Chlamydia pneumoniae
External Id: CHEMBL1286501
Name: Antileishmanial activity against axenic amastigote Leishmania donovani MHOM/SD/1962/1...
Source: ChEMBL
Target: Leishmania donovani
External Id: CHEMBL3406136
Name: Cytotoxicity against human HL cells assessed as cell viability at 10 uM after 72 hrs ...
Source: ChEMBL
Target: HL
External Id: CHEMBL1286502
Name: Antibacterial activity against Chlamydia pneumoniae CWL029 infected in human HL cells...
Source: ChEMBL
Target: Chlamydia pneumoniae
External Id: CHEMBL1286504
Name: Cytotoxicity against human HL cells at 2.5 uM after 72 hrs by celltiter-glo analysis
Source: ChEMBL
Target: HL
External Id: CHEMBL1286507
Name: Antibacterial activity against Staphylococcus aureus ATCC 25923 assessed as inhibitio...
Source: ChEMBL
Target: Staphylococcus aureus
External Id: CHEMBL1286508
Name: Antibacterial activity against Escherichia coli ATCC 25922 assessed as inhibition of ...
Source: ChEMBL
Target: Escherichia coli
External Id: CHEMBL1286509
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