ARC-239
Modify Date: 2024-01-10 17:47:08
ARC-239 structure
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Common Name | ARC-239 | ||
|---|---|---|---|---|
| CAS Number | 67339-62-2 | Molecular Weight | 407.51 | |
| Density | 1.167g/cm3 | Boiling Point | 595.8ºC at 760 mmHg | |
| Molecular Formula | C24H29N3O3 | Melting Point | N/A | |
| MSDS | Chinese USA | Flash Point | 314.1ºC | |
Use of ARC-239ARC 239 is an α2B/C-adrenergic receptor antagonist with pKi of 7.06 and 6.95 for rat kidney α2B and human α2C, respectively. ARC 239 also inhibits 5-HT1A receptor with a Ki of 63.1 nM[1][2]. |
| Name | ARC 239 dihydrochloride hydrate |
|---|---|
| Synonym | More Synonyms |
| Description | ARC 239 is an α2B/C-adrenergic receptor antagonist with pKi of 7.06 and 6.95 for rat kidney α2B and human α2C, respectively. ARC 239 also inhibits 5-HT1A receptor with a Ki of 63.1 nM[1][2]. |
|---|---|
| Related Catalog | |
| Target |
human α2C-adrenoceptor:6.95 (pKi) Alpha-2C adrenergic receptor:7.06 (pKi) 5-HT1A Receptor:63.1 nM (Ki) |
| References |
| Density | 1.167g/cm3 |
|---|---|
| Boiling Point | 595.8ºC at 760 mmHg |
| Molecular Formula | C24H29N3O3 |
| Molecular Weight | 407.51 |
| Flash Point | 314.1ºC |
| Exact Mass | 479.17400 |
| PSA | 53.09000 |
| LogP | 4.32220 |
| Index of Refraction | 1.576 |
| ARC 239 dihydrochloride,2-[2-(4-(2-Methoxyphenyl)piperazin-1-yl)ethyl]-4,4-dimethyl-1,3-(2H,4H)-isoquinolindionedihydrochloride |