α-Helical CRF(9-41) structure
|
Common Name | α-Helical CRF(9-41) | ||
|---|---|---|---|---|
| CAS Number | 90880-23-2 | Molecular Weight | 3826.40 | |
| Density | N/A | Boiling Point | N/A | |
| Molecular Formula | C166H274N46O53S2 | Melting Point | N/A | |
| MSDS | N/A | Flash Point | N/A | |
Use of α-Helical CRF(9-41)α-Helical CRF(9-41) is a competitive CRF2 receptor antagonist with KB of ~100 nM. α-Helical CRF(9-41) is also a partial agonist of CRF1 receptor with an EC50 of 140 nM[1][2]. |
| Name | α-Helical CRF(9-41) |
|---|
| Description | α-Helical CRF(9-41) is a competitive CRF2 receptor antagonist with KB of ~100 nM. α-Helical CRF(9-41) is also a partial agonist of CRF1 receptor with an EC50 of 140 nM[1][2]. |
|---|---|
| Related Catalog | |
| Target |
KB: ~100 nM (CRF2 receptor)[2] EC50: 140 nM (CRF1 receptor)[2] |
| References |
| Molecular Formula | C166H274N46O53S2 |
|---|---|
| Molecular Weight | 3826.40 |