Synlett

General and Easy Access to 11-Substituted 4-Hydroxy-2, 3, 4, 5-tetrahydro [1, 4] diazepino [1, 2-a] indol-1-one Derivatives

A Putey, G Fournet, B Joseph

Index: Synlett, , # 17 p. 2755 - 2758

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Citation Number: 3

Abstract

... Synlett 2006(17): 2755-2758 DOI: 10.1055/s-2006-950249. ... Treatment of commercially available p-anisaldehyde with ethyl azidoacetate in the presence of MeONa yielded the azidoacrylate, which was converted into indole 1c by refluxing in xylene (overall yield 68%). ...

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