Tetrahedron

Oxidation of indoles and 1, 2-dihydro-3H-indol-3-ones

E Desarbre, L Savelon, O Cornec, JY Merour

Index: Desarbre; Savelon; Cornec; Merour Tetrahedron, 1996 , vol. 52, # 8 p. 2983 - 2994

Full Text: HTML

Citation Number: 8

Abstract

2-Hydroxy-1, 2-dihydro-3H-indol-3-ones 3 were obtained from 1, 2-dihydro-3H-indol-3-ones 2 by using various conditions (m-CPBA or sodium azide) depending on substituent in 1- position. The reactivity of hydroxyketones 3 is examined and oxidation of 1-(phenylsulfonyl) indole by m-CPBA is described.

Related Articles:

1-Acetyl-2-bromo-3-indolinone in nucleophilic substitution reactions and the synthesis of pyrrolo [3, 2-b] indoles

[Velezheva, V. S.; Mel'man, A. I.; Smushkevich, Yu. I.; Pol'shakov, V. I.; Anisimova, O. S. Pharmaceutical Chemistry Journal, 1990 , vol. 24, # 12 p. 917 - 923 Khimiko-Farmatsevticheskii Zhurnal, 1990 , vol. 24, # 12 p. 46 - 51]

Total synthesis of (+)-isatisine A

[Kawasaki, Tomomi; Chien, Chun-Sheng; Suzuki, Takako; Takanami, Toshikatsu; Sakamoto, Masanori Heterocycles, 1985 , vol. 23, # 1 p. 172]

More Articles...