Elemental fluorine. Part 5. Reactions of 1, 3-dithiolanes and thioglycosides with fluorine–iodine mixtures
RD Chambers, G Sandford, ME Sparrowhawk…
Index: Chambers, Richard D.; Sandford, Graham; Sparrowhawk, Matthew E.; Atherton, Malcolm J. Journal of the Chemical Society - Perkin Transactions 1, 1996 , # 16 p. 1941 - 1944
Full Text: HTML
Citation Number: 0
Abstract
1, 3-Dithiolanes, prepared from diaryl ketones, react with elemental fluorine–iodine mixtures to give the corresponding difluoromethylene derivatives. Under the same conditions, thioglycosides give glycosyl fluorides in good yields. Reaction of 1, 3-dithiolanes with fluorine in aqueous acetonitrile provides a remarkably mild method for efficient deprotection to the parent ketone.
Related Articles:
[Ten Brink, Gerd-Jan; Arends, Isabel W. C. E.; Hoogenraad, Marcel; Verspui, Goeran; Sheldon, Roger A. Advanced Synthesis and Catalysis, 2003 , vol. 345, # 12 p. 1341 - 1352]
[Angewandte Chemie - International Edition, , vol. 41, # 23 p. 4563 - 4565]
[Journal of the American Chemical Society, , vol. 108, p. 536 - 538]
[Fort, Y.; Vanderesse, R.; Caubere, P. Chemistry Letters, 1988 , # 5 p. 757 - 760]
[Lou, Ji-Dong; Lin, Fang; Lu, Xiu Lian; Wang, Qiang; Zou, Xiao-Nan Synthesis and Reactivity in Inorganic, Metal-Organic and Nano-Metal Chemistry, 2012 , vol. 42, # 2 p. 282 - 284]