Tetrahedron Letters

Regioselective methylation of indazoles using methyl 2, 2, 2-trichloromethylacetimidate

SR Baddam, NU Kumar, AP Reddy, R Bandichhor

Index: Tetrahedron Letters, , vol. 54, # 13 p. 1661 - 1663

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Citation Number: 5

Abstract

... Tetrahedron Letters. Volume 54, Issue 13, 27 March 2013, Pages 1661–1663. ... These screening efforts reveal that 2.5 equiv is the optimum quantity for regioselective methylation of 7 (a–k). The quantity of solvent, dichloromethane was adjudged to be 25 vol with respect to ...

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