Extending the Scope of the Aza??Fischer Synthesis of 4??and 6??Azaindoles

…, J Coste, G Guillaumet, F Suzenet

Index: Thomae, David; Jeanty, Matthieu; Coste, Jerome; Guillaumet, Gerald; Suzenet, Franck European Journal of Organic Chemistry, 2013 , # 16 p. 3328 - 3336

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Abstract

Abstract Fischer indole cyclization has recently been described as an efficient approach to the synthesis of azaindoles bearing electron-donating groups. We now show that this cascade reaction can be very efficient for the formation of a wider range of 4-and 6- ...

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