Efficient synthesis of a 7-azabicyclo [2.2. 1] heptane based GlyT1 uptake inhibitor

H Xiong, W Frietze, DW Andisik, GE Ernst, WE Palmer…

Index: Xiong, Hui; Frietze, William; Andisik, Donald W.; Ernst, Glen E.; Palmer, William E.; Hinkley, Lindsay; Varnes, Jeffrey G.; Albert, Jeffrey S.; Veale, Chris A. Tetrahedron Letters, 2010 , vol. 51, # 51 p. 6741 - 6744

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Citation Number: 5

Abstract

Download PDF Opens in a new window. Article suggestions will be shown in a dialog on return to ScienceDirect. ... Please enable JavaScript to use all the features on this page. ... An efficient synthetic route based on generation and subsequent electrophilic reaction of a Boc-protected azabicyclo[2.2.1]heptane anion to prepare a potent GlyT1 uptake inhibitor (1) is described. ... Generation and subsequent electrophilic reaction of a Boc-protected azabicyclo[2.2.1] ...