Identification of a novel series of tetrahydrodibenzazocines as inhibitors of 17β-hydroxysteroid dehydrogenase type 3

BE Fink, AV Gavai, JS Tokarski, B Goyal…

Index: Bioorganic and Medicinal Chemistry Letters, , vol. 16, # 6 p. 1532 - 1536

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Citation Number: 30

Abstract

... Please enable JavaScript to use all the features on this page. Bioorganic & Medicinal Chemistry Letters. ... 8 The dibenzothiazocine 1 9 represented an attractive starting point for medicinal chemistry, based on its potency in the biochemical and cell-based assays. ...

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