Tetrahedron Letters

A facile access to substituted indoles utilizing palladium catalyzed annulation under microwave enhanced conditions

…, KR Haridas, AM Sajith, A Muralidharan

Index: Karuvalam, Ranjith P.; Haridas, Karickal R.; Sajith, Ayyiliath M.; Muralidharan, Arayambath Tetrahedron Letters, 2013 , vol. 54, # 37 p. 5126 - 5129

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Citation Number: 4

Abstract

Abstract A facile access to differently substituted indoles using palladium catalyzed annulation reactions under microwave enhanced conditions has been achieved. A highly active and efficient catalytic system PdCl 2/(A-taphos) for the synthesis of indole via palladium catalyzed ring annulation of ortho iodo anilines and aldehydes has been developed.

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