A novel type of retinoic acid receptor antagonist: synthesis and structure-activity relationships of heterocyclic ring-containing benzoic acid derivatives

H Yoshimura, M Nagai, S Hibi, K Kikuchi…

Index: Journal of Medicinal Chemistry, , vol. 38, # 16 p. 3163 - 3173

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Citation Number: 49

Abstract

... Instead of showing agonism, as did compound 2, it was antagonistic to ATRA in the HL-60 assay. It should be 0 1995 American Chemical Society Page 2. 3164 Journal of Medicinal Chemistry, 1995, Vol. 38, No. 16 Chart 1 Yoshimura et al. HN-N HN-N ...