Development of an Acyl Sulfonamide Anti-Proliferative Agent, LY573636· Na†

MH Yates, NJ Kallman, CP Ley…

Index: Sone, Tyo; Abe, Yukio; Sato, Norio; Ebina, Manabu Bulletin of the Chemical Society of Japan, 1985 , vol. 58, # 3 p. 1063 - 1064

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Abstract

... Initial supplies were met using the chemistry outlined in Scheme 1. figure Scheme 1. Initial synthesis of ... 2.1 Preparation of Sulfonyl Chloride 2 2-Bromothiophene 1 is a bulk commodity chemical which can be processed under well established conditions(2) to give the ...

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