Palladium/tetraphosphine catalyzed suzuki cross??coupling of heteroarylboronic acids with aryl halides

I Kondolff, H Doucet, M Santelli

Index: Kondolff, Isabelle; Doucet, Henri; Santelli, Maurice Journal of Heterocyclic Chemistry, 2008 , vol. 45, # 1 p. 109 - 118

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Citation Number: 22

Abstract

Due to their important biological properties, the preparation of heterobiaryls is an important industrial goal. The palladium-catalysed Suzuki cross-coupling reaction between heteroaryl halides and arylboronic acids provides a very efficient method for the preparation of heterobiaryl derivatives [1, 2]. On the other hand, the reverse reaction using heteroarylboronic acids and aryl halides has attracted much less attention, and most of the ...