Tetrahedron letters

One pot conversion of azido arenes to N-arylacetamides and N-arylformamides: synthesis of 1, 4-benzodiazepine-2, 5-diones and fused [2, 1-b] quinazolinones

A Kamal, AV Ramana, KS Reddy, KV Ramana…

Index: Kamal, Ahmed; Ramana, A. Venkata; Reddy, K. Srinivasa; Ramana, K. Venkata; Hari Babu; Prasad, B. Rajendra Tetrahedron Letters, 2004 , vol. 45, # 44 p. 8187 - 8190

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Citation Number: 31

Abstract

Sodium iodide in acidic media has been employed for the synthesis of N-arylformamides and N-arylacetamides. The NaI/acetic acid reagent system has also been extended for the synthesis of 1, 4-benzodiazepine-2, 5-diones, pyrrolo [2, 1-c][1, 4] benzodiazepine-5, 11- diones, and fused [2, 1-b] quinazolinones.

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