Optimization of the aromatase inhibitory activities of pyridylthiazole analogues of resveratrol

AS Mayhoub, L Marler, TP Kondratyuk, EJ Park…

Index: Bioorganic and Medicinal Chemistry, , vol. 20, # 7 p. 2427 - 2434

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Citation Number: 18

Abstract

... Bioorganic & Medicinal Chemistry. ... a Department of Medicinal Chemistry and Molecular Pharmacology ... 17 Further chemical optimization of the lead compound 2 furnished 3,5-dipyridyl-1,2,4-thiadiazoles (eg, compound 3) as a new class of non-steroidal aromatase ...

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