Synthesis and pharmacological activity of partially modified retro-inverso dermorphin tetrapeptides

S Salvadori, M Marastoni, G Balboni…

Index: Salvadori, Severo; Marastoni, Mauro; Balboni, Gianfranco; Sarto, Gian Pietro; Tomatis, Roberto Journal of Medicinal Chemistry, 1985 , vol. 28, # 6 p. 769 - 774

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Citation Number: 16

Abstract

Severo Salvadori,t Mauro Marastoni,f Gianfranco Balboni,* Gian Pietro Sarto,s and Roberto Tomatis*$ ... Institute of Pharmaceutical Chemistry and Institute of Pharmacology, University of Ferrara, 44100 Ferrara, Italy. Received April 23, 1984 ... We studied the effect of partial retro-inverso modification of selected peptide bonds of N-terminal tetrapeptide analogues of dermorphin (H-Tyr-D-Ala-Phe-Gly-Tyr-Pro-Ser-NHJ. ... Dermorphins are opioid ...

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