Discovery of new C3aR ligands. Part 2: Amino-piperidine derivatives

F Denonne, S Binet, M Burton, P Collart…

Index: Bioorganic and Medicinal Chemistry Letters, , vol. 17, # 12 p. 3262 - 3265

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Citation Number: 11

Abstract

... Bioorganic & Medicinal Chemistry Letters. ... Compound 5 in particular was quite attractive to start a medicinal chemistry program as it had much better solubility than the starting hit (0.1 mg/ml instead of <0.0001 mg/ml). ...

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