Synthesis and pharmacological activity of benzo [b] thiophene??3??carboxylic acid derivatives

A Shafiee, MA Hedayati, MM Salimi…

Index: Shafiee; Hedayati; Salimi; Faghihi Journal of Pharmaceutical Sciences, 1983 , vol. 72, # 2 p. 198 - 202

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Citation Number: 3

Abstract

Abstract Several dialkylaminoethyl benzo [b] thiophene-3-carboxylates, N-(2- dialkylaminoethyl) benzo [b] thiophene-3-carboxamides, 2-dialkylaminoethyl benzo [b] thiophene-3-carbamates, and substituted ureas with benzo [b] thiophene moiety, were prepared and tested for local anesthetic, anticholinergic, and antihistaminic activities. Several of the compounds showed significant activity.

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