Tetrahedron

Convenient synthesis of C-terminal di-and tri-peptide amides from N-protected dipeptidoylbenzotriazoles

I Celik, AAA Abdel-Fattah

Index: Celik, Ilhami; Abdel-Fattah, Ashraf A.A. Tetrahedron, 2009 , vol. 65, # 25 p. 4923 - 4929

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Citation Number: 3

Abstract

Download PDF Opens in a new window. Article suggestions will be shown in a dialog on return to ScienceDirect. ... Please enable JavaScript to use all the features on this page. ... N-Protected dipeptidoylbenzotriazoles react with aqueous ammonia to give dipeptide primary amides (77–98%) and with N-unprotected α-amino amides to afford tripeptide primary amides (82–86%). ... Chemical structures of the aspartyl protease inhibitors l-682,679 and ...

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