Synthesis and biological evaluation of novel irreversible serine protease inhibitors using amino acid based sulfonyl fluorides as an electrophilic trap

AJ Brouwer, T Ceylan, AM Jonker…

Index: Bioorganic and Medicinal Chemistry, , vol. 19, # 7 p. 2397 - 2406

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Citation Number: 15

Abstract

... Bioorganic & Medicinal Chemistry. ... Department of Medicinal Chemistry and Chemical Biology, Utrecht Institute for Pharmaceutical Sciences, Faculty of Science, Utrecht University, PO Box 80082, 3508 TB Utrecht, The Netherlands. ...

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