Benzannulation from Alkyne without Metallic Catalysts at Room Temperature to 100° C
T Jin, F Yang, Y Yamamoto
Index: Jin, Tienan; Yang, Fan; Yamamoto, Yoshinori Organic Letters, 2010 , vol. 12, # 2 p. 388 - 390
Full Text: HTML
Citation Number: 13
Abstract
An efficient, novel metal-catalyst-free aminobenzannulation of 2-(prop-2-ynyl)(oxo) benzenes 1 with various dialkylamines 2 afforded a variety of 2-aminonaphthalenes 3 in good to excellent yields under mild reaction conditions at room temperature to 100° C (at most).
Related Articles:
[Zhou, Yanping; Xie, Yinjun; Yang, Lei; Xie, Pan; Huang, Hanmin Tetrahedron Letters, 2013 , vol. 54, # 21 p. 2713 - 2716]
[Tobisu, Mamoru; Shimasaki, Toshiaki; Chatani, Naoto Chemistry Letters, 2009 , vol. 38, # 7 p. 710 - 711]
[Ramgren, Stephen D.; Silberstein, Amanda L.; Yang, Yang; Garg, Neil K. Angewandte Chemie - International Edition, 2011 , vol. 50, # 9 p. 2171 - 2173]
[Carmack, Marvin; Behforouz, Mohammad; Berchtold, Glenn A.; Berkowitz, Samuel M.; Wiesler, Donald; Barone, Ralph Journal of Heterocyclic Chemistry, 1989 , vol. 26, p. 1305 - 1318]