Synthesis of di-and tripeptide analogues containing α-ketoamide as a new core structure for inhibition of HIV-1 protease

MM Sheha, NM Mahfouz, HY Hassan…

Index: European Journal of Medicinal Chemistry, , vol. 35, # 10 p. 887 - 894

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Citation Number: 52

Abstract

... European Journal of Medicinal Chemistry. ... b Pharmaceutical & Biotechnology Laboratory, Japan Energy Co., Kyoto, Japan; c Department of Medicinal Chemistry Kyoto Pharmaceutical University, Yamashinaku ... 1 H-NMR (DMSO-d 6 ) δ: 1.27, (s, 9H), 2.64 (d, 2H, J=8.3 Hz), 3.37 (bs ...

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